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Journal articles
Synthesis of Bridged Tetrahydrobenzo[b]azepines and Derivatives through an Aza-Piancatelli Cyclization/Michael Addition Sequence
Abstract : Herein, we report the preparation of bridged tetrahydrobenzo[b]azepines, which was accomplished through an aza-Piancatelli cyclization/Michael addition sequence in a one-pot fashion from readily available precursors. It is noteworthy that a general method to access these scaffolds was hitherto unprecedented. Additionally, the multifaceted aspects of this process have been exemplified through its application to the synthesis of 2-azabicyclo[3.2.1]octanes and bridged tetrahydrobenzo[b]oxepines, along with post-derivatizations.
Cited literature [31 references]
https://hal-univ-rennes1.archives-ouvertes.fr/hal-02438534
Contributor : Laurent Jonchère <>
Submitted on : Tuesday, February 11, 2020 - 4:40:33 PM
Last modification on : Saturday, October 3, 2020 - 4:15:43 AM
Long-term archiving on: : Tuesday, May 12, 2020 - 4:28:39 PM
Contributor : Laurent Jonchère <>
Submitted on : Tuesday, February 11, 2020 - 4:40:33 PM
Last modification on : Saturday, October 3, 2020 - 4:15:43 AM
Long-term archiving on: : Tuesday, May 12, 2020 - 4:28:39 PM
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Wang et al-Synthesis of Bridge...
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